SCHEMBL28069972

SCHEMBL28069972

ClCCOc1ccc2c(NOCCCc3ccccc3)ncnc2c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.47
AURKA O14965 8/20 0.44
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
DNMT1 P26358 4/20 0.42
DNMT3A Q9Y6K1 4/20 0.42
PIK3CD O00329 1/20 0.42
PIK3R1 P27986 1/20 0.42
AURKB Q96GD4 7/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
KDR P35968 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK1 P28482 2/20 0.40
LMNA P02545 1/20 0.40
APP P05067 1/20 0.40
HTT P42858 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16586076 0.86 PIK3CD (0.58) EGFRAURKADNMT1DNMT3APIK3CD
SCHEMBL16596382 0.82 PIK3CD (0.60) EGFRAURKADNMT1DNMT3APIK3CD
SCHEMBL28049941 0.78 MAOA (0.50) EGFRAURKAMAOAMAOBPIK3CD
SCHEMBL17994857 0.76 EGFR (0.61) EGFRAURKADNMT1DNMT3APIK3CD
SCHEMBL12694408 0.76 EGFR (0.68) EGFRAURKAAURKBKDR
SCHEMBL17994858 0.74 EGFR (0.58) EGFRAURKADNMT1DNMT3APIK3CD
SCHEMBL19563559 0.72 AURKA (0.51) EGFRAURKADNMT1DNMT3APIK3CD
SCHEMBL1938919 0.70 AURKA (0.54) EGFRAURKADNMT1DNMT3AMEN1
SCHEMBL27969044 0.70 MAOA (0.50) MAOAMAOBMEN1MAPTKMT2A
SCHEMBL1939067 0.70 AURKA (0.81) AURKAAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105555781-A Quinazoline derivatives and their use as DNA methyltransferase inhibitors PF MEDICAMENT 2016-05-04 CN disclosed