SCHEMBL28070960

SCHEMBL28070960

CC(C)(C)OC(=O)N1CCC(n2cc(-c3ccccc3)nn2)CC1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.53
DRD4 P21917 1/20 0.53
DRD3 P35462 1/20 0.53
GPR119 Q8TDV5 5/20 0.51
USP30 Q70CQ3 5/20 0.50
KDM5C P41229 2/20 0.50
KDM2A Q9Y2K7 2/20 0.50
KDM3A Q9Y4C1 1/20 0.50
KDM6B O15054 1/20 0.49
KDM4A O75164 1/20 0.49
KDM4C Q9H3R0 1/20 0.49
KDM4E B2RXH2 1/20 0.49
PKM P14618 1/20 0.49
EGFR P00533 1/20 0.48
SRC P12931 1/20 0.48
HPGDS O60760 1/20 0.47
GRM5 P41594 1/20 0.47
GRM1 Q13255 1/20 0.47
ABHD6 Q9BV23 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22712368 0.89 GRM5 (0.48) GPR119KDM5CKDM2AKDM3AGRM5
SCHEMBL31260529 0.89 PIK3CA (0.47) GPR119KDM5CKDM2AKDM3ASRC
SCHEMBL1781995 0.83 USP30 (0.53) GPR119USP30KDM4EPKMEGFR
SCHEMBL2225927 0.81 KDM5C (0.44) GPR119KDM5CKDM2AKDM3AKDM6B
SCHEMBL14692527 0.81 GPR119 (0.46) GPR119KDM5CKDM2AKDM3AKDM4E
SCHEMBL22730550 0.81 DDB1 (0.48) GPR119KDM5CKDM2AKDM3AKDM4E
SCHEMBL18376153 0.81 GPR119 (0.47) GPR119KDM5CKDM2AKDM3AKDM4E
SCHEMBL1653749 0.81 TNK2 (0.56) GPR119USP30EGFRSRCHPGDS
SCHEMBL18367623 0.80 GPR119 (0.46) GPR119KDM4EPKM
SCHEMBL16716871 0.80 GPR119 (0.46) GPR119KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646492-A Five-membered-aromatic-heterocycte-containing substituted xanthine compound and preparation method and use thereof 中国医学科学院药物研究所 2016-06-08 CN disclosed