SCHEMBL28071072

SCHEMBL28071072

FC(F)C(F)c1cccnc1N1CCNCC1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.56
HTR2C P28335 4/20 0.47
PLD1 Q13393 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HTR2A P28223 1/20 0.43
SLC6A4 P31645 1/20 0.43
HTR3E A5X5Y0 1/20 0.42
HTR3B O95264 1/20 0.42
HTR1A P08908 1/20 0.42
HTR3A P46098 1/20 0.42
HTR3D Q70Z44 1/20 0.42
HTR3C Q8WXA8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19107153 0.81 EPHX2 (0.55) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL6111507 0.79 EPHX2 (0.52) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL19853561 0.77 EPHX2 (0.50) EPHX2HTR2CPLD1
SCHEMBL1758382 0.76 EPHX2 (0.64) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL9078264 0.75 EPHX2 (0.49) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL28082095 0.75 EPHX2 (0.49) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL31651713 0.75 EPHX2 (0.55) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL18842836 0.74 EPHX2 (0.48) EPHX2HTR2CPLD1
Hydrochloric Acid SCHEMBL10960670 0.74 EPHX2 (0.62) EPHX2HTR2CPLD1KDM4EALDH1A1
SCHEMBL10495676 0.74 HTR2C (0.68) EPHX2HTR2CPLD1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104470924-B Imidazopyrazines derivant as TNF active regulator UCB生物制药私人有限公司 2016-11-09 CN disclosed
CN-105814051-A Tetrahydroimidazopyridine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed