SCHEMBL28072026

SCHEMBL28072026

COc1ccc(C(O)Cc2ccccn2)cc1OC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.53
HTT P42858 1/20 0.53
ALDH1A1 P00352 7/20 0.48
KMT2A Q03164 4/20 0.48
MEN1 O00255 3/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C19 P33261 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
ALOX15 P16050 1/20 0.48
ACHE P22303 1/20 0.47
HIF1A Q16665 1/20 0.46
EPAS1 Q99814 1/20 0.46
KDM4E B2RXH2 3/20 0.46
PPARG P37231 1/20 0.46
PPARD Q03181 1/20 0.46
PPARA Q07869 1/20 0.46
NFKB1 P19838 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPT P10636 1/20 0.44
BLM P54132 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28162053 0.90 TP53 (0.45) TP53HTTALDH1A1KMT2AMEN1
SCHEMBL7321974 0.86 PDE4A (0.61) PDE4APDE4BPDE4CPDE4D
SCHEMBL11084913 0.81 MEN1 (0.50) ALDH1A1KMT2AMEN1KDM4EMAPT
SCHEMBL7042336 0.79 TP53 (0.56) TP53HTTKMT2AACHEHIF1A
SCHEMBL7389132 0.77 PDE4A (0.49) ALDH1A1KMT2AMEN1CYP1A2CYP2C19
SCHEMBL28162614 0.77 PTPRA (0.40) KMT2AMEN1CYP1A2CYP2C19KDM4E
SCHEMBL6583680 0.76 PDE4B (0.42) TP53HTTALDH1A1KMT2AMEN1
SCHEMBL23610053 0.75 ACHE (0.53) TP53HTTKMT2AMEN1CYP1A2
SCHEMBL31143787 0.75 ACHE (0.53) TP53HTTKMT2AMEN1CYP1A2
SCHEMBL11619843 0.75 ACHE (0.53) TP53HTTKMT2AMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104837828-B It is used as the phenylethyl pyridine derivate of PDE4 inhibitor 奇斯药制品公司 2017-07-18 CN disclosed
CN-105814034-A Benzhydryl derivatives for the treatment of respiratory diseases 奇斯药制品公司 2016-07-27 CN disclosed
CN-105793250-A Heteroaryl derivatives for the treatment of respiratory diseases 奇斯药制品公司 2016-07-20 CN disclosed