SCHEMBL28072259

SCHEMBL28072259

O=C(O)c1cnc2ccc(Nc3ccc(C(F)(F)F)cc3)cc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.48
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 2/20 0.45
AURKA O14965 1/20 0.45
DHFR P00374 1/20 0.43
EPHX2 P34913 1/20 0.43
PIN1 Q13526 1/20 0.42
TRPV1 Q8NER1 3/20 0.42
ABCG2 Q9UNQ0 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
MAPT P10636 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
CSF1R P07333 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10474372 0.85 MGAM (0.57) MGAMSRD5A2
SCHEMBL18372036 0.76 SMN1; SMN2 (0.49) MGAMNPC1RAB9ASRD5A2
SCHEMBL22376 0.76 MGAM (0.57) MGAMSRD5A2
SCHEMBL5447688 0.75 SRD5A2 (0.69) AKR1C3AKR1C2EPHX2TRPV1NPC1
SCHEMBL1352938 0.74 HDAC6 (0.57) MGAM
SCHEMBL10465639 0.74 MGAM (0.70) MGAMNPC1RAB9AMEN1KMT2A
SCHEMBL13279924 0.74 AKR1C3 (0.78) AKR1C3AKR1C2AURKAEPHX2NPC1
SCHEMBL1644022 0.74 MGAM (0.57) MGAMEPHX2TRPV1SRD5A2
SCHEMBL12133241 0.73 ALOX15 (0.50) MGAMABCG2NPC1RAB9AMEN1
SCHEMBL12133496 0.73 HDAC6 (0.48) NPC1RAB9APOLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105722840-B fused quinoline compound as PI3K, mTOR inhibitors 杭州爱德程医药科技有限公司 2018-01-05 CN disclosed
CN-105722840-A Fused quinoline compunds as PI3K, mTOR inhibitors 杭州爱德程医药科技有限公司 2016-06-29 CN disclosed