SCHEMBL28073276

SCHEMBL28073276

CCC(C)C(NC(=O)C(O)(NC(=O)CCCc1ccccc1)C(C)(C)N)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.51
MAPK1 P28482 1/20 0.45
HPGD P15428 1/20 0.44
LMNA P02545 1/20 0.42
PKM P14618 1/20 0.42
EPHX2 P34913 2/20 0.41
HDAC1 Q13547 2/20 0.40
HDAC3 O15379 1/20 0.40
HDAC2 Q92769 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
HDAC5 Q9UQL6 1/20 0.40
KMT2A Q03164 3/20 0.40
MEN1 O00255 2/20 0.40
ANPEP P15144 1/20 0.39
ATM Q13315 1/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15411973 1.00 SMN1; SMN2 (0.51) SMN1; SMN2MAPK1HPGDLMNAPKM
SCHEMBL21570179 0.82 HDAC1 (0.53) SMN1; SMN2MAPK1HPGDLMNAPKM
SCHEMBL5808627 0.82 HDAC1 (0.53) SMN1; SMN2MAPK1HPGDLMNAPKM
SCHEMBL5819414 0.77 SMN1; SMN2 (0.52) SMN1; SMN2MAPK1HPGDLMNAPKM
SCHEMBL8089676 0.74 SMN1; SMN2 (0.57) SMN1; SMN2MAPK1HPGDEPHX2HDAC3
SCHEMBL8085372 0.74 SMN1; SMN2 (0.57) SMN1; SMN2MAPK1HPGDEPHX2HDAC3
SCHEMBL12807096 0.73 KMT2A (0.47) MAPK1KMT2AMEN1ANPEPATM
SCHEMBL17867024 0.73 PLA2G2A (0.35) SMN1; SMN2EPHX2
SCHEMBL12807097 0.73 KMT2A (0.47) MAPK1KMT2AMEN1ANPEPATM
SCHEMBL27860159 0.73 KMT2A (0.47) MAPK1KMT2AMEN1ANPEPATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105985405-A 3-amino-2-hydroxy-4-phenyl-valyl-isoleucine derivative and application thereof 上海来益生物药物研究开发中心有限责任公司 2016-10-05 CN disclosed
CN-105001301-A 3-amino-2-hydroxy-4-phenyl-valyl-isoleucine synthesis method SHANGHAI LAIYI BIOMEDICAL RES AND DEV CT CO LTD 2015-10-28 CN disclosed