SCHEMBL28075560

SCHEMBL28075560

COc1ccc(-c2nc(-c3ccc(OC)c([N+](=O)[O-])c3)n[nH]2)cc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 1/20 0.55
LMNA P02545 4/20 0.50
ALDH1A1 P00352 1/20 0.50
NR1H2 P55055 1/20 0.50
NR1H3 Q13133 1/20 0.50
PDGFRB P09619 1/20 0.50
PDGFRA P16234 1/20 0.50
MAPT P10636 4/20 0.46
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 2/20 0.45
POLB P06746 1/20 0.45
ADORA2A P29274 1/20 0.45
ADORA1 P30542 1/20 0.45
NPC1 O15118 1/20 0.45
NFKB1 P19838 1/20 0.45
MAPK1 P28482 1/20 0.45
STAT1 P42224 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28075509 0.90 GRK6 (0.60) GRK6LMNAALDH1A1PDGFRBPDGFRA
SCHEMBL28075506 0.89 NR1H2 (0.61) GRK6LMNAALDH1A1NR1H2NR1H3
SCHEMBL28075564 0.87 GRK6 (0.54) GRK6LMNAALDH1A1PDGFRBPDGFRA
SCHEMBL4680875 0.83 GRK6 (0.53) GRK6
SCHEMBL28075567 0.83 GRK6 (0.50) GRK6LMNAALDH1A1PDGFRBPDGFRA
SCHEMBL28075557 0.82 GRK6 (0.52) GRK6LMNAALDH1A1PDGFRBPDGFRA
SCHEMBL19356065 0.81 PDGFRB (0.53) GRK6LMNAALDH1A1PDGFRBPDGFRA
SCHEMBL12312144 0.79 PDGFRB (0.57) LMNAALDH1A1PDGFRBPDGFRAMAPT
SCHEMBL28075511 0.79 KDM4E (0.58) LMNAALDH1A1NR1H2NR1H3MAPT
SCHEMBL15117068 0.77 KDM4E (0.67) LMNAALDH1A1NR1H2NR1H3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN claimed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN claimed
CN-106008557-B 3,6- diaryl-[1,2,4] triazole simultaneously purposes of [3,4-b] [1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2019-03-01 CN disclosed
CN-106008557-A Application of 3,6-diaryl-[1,2,4] triazolo[3,4-b][1,3,4] thiadiazole compound as tumor cell proliferation inhibitor 沈阳药科大学 2016-10-12 CN disclosed