SCHEMBL28075992

SCHEMBL28075992

N#Cc1ccc(B(O)OCl)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.59
CA2 P00918 4/20 0.43
CA9 Q16790 2/20 0.43
CA12 O43570 1/20 0.43
CA3 P07451 1/20 0.43
CA6 P23280 1/20 0.43
CA14 Q9ULX7 1/20 0.43
MMP3 P08254 1/20 0.39
CYP2A6 P11509 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CA1 P00915 3/20 0.36
CYP19A1 P11511 1/20 0.36
TSHR P16473 2/20 0.36
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27532994 0.79 ENPP2 (0.59) ENPP2CA2CA9CA12CA3
SCHEMBL21133795 0.79 ENPP2 (0.59) ENPP2CA2CA9CA12CA3
SCHEMBL1820855 0.77 ENPP2 (0.65) ENPP2ALDH1A1TSHRMAPTGSK3B
SCHEMBL23797214 0.76 ENPP2 (0.55) ENPP2CA2CA9CA12CA3
SCHEMBL2405727 0.75 ENPP2 (0.73) ENPP2CA2CA9CA12CA3
SCHEMBL6016 0.75 ENPP2 (1.00) ENPP2CA2CA9CA12CA3
SCHEMBL20975981 0.75 ENPP2 (0.53) ENPP2CA2CA9CA12CA3
SCHEMBL14421551 0.74 ENPP2 (0.64) ENPP2CA2CA9CA12CA3
SCHEMBL1138376 0.73 ENPP2 (0.52) ENPP2CA2CA9CA12CA3
SCHEMBL21336582 0.71 ENPP2 (0.67) ENPP2CA2CA9CA12CA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106488921-B Aldosterone synthase inhibitors 勃林格殷格翰国际有限公司 2019-03-15 CN disclosed
CN-107406433-A Derivatives of 2, 3-diphenylchromene for the treatment of cancer 豪夫迈·罗氏有限公司 2017-11-28 CN disclosed
CN-103958487-B Benzoic acid derivative as EIF4E inhibitor 霍夫曼-拉罗奇有限公司 2016-07-13 CN disclosed