SCHEMBL28076643

SCHEMBL28076643

COc1ccc(N)c(CCBr)c1CCBr

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.46
EP300 Q09472 1/20 0.44
KAT8 Q9H7Z6 1/20 0.44
ALDH1A1 P00352 8/20 0.40
GAA P10253 1/20 0.40
CYP3A4 P08684 3/20 0.39
TDP1 Q9NUW8 3/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 2/20 0.39
THRB P10828 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
FGB P02675 1/20 0.39
MAPK1 P28482 1/20 0.39
ADORA2A P29274 1/20 0.39
PPARG P37231 1/20 0.39
RAB9A P51151 1/20 0.39
NCOA2 Q15596 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28290607 0.82 IDO1 (0.47) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL9382243 0.82 IDO1 (0.47) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL28468316 0.79 SKP2 (0.44) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL9317755 0.75 CA1 (0.46) ALDH1A1CYP3A4TDP1TSHRHSD17B10
SCHEMBL28207495 0.74 IDO1 (0.45) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL27354250 0.70 ERN1 (0.45) ALDH1A1TDP1TSHRMAPTRAB9A
SCHEMBL5142101 0.69 CA2 (0.41) IDO1ALDH1A1GAACYP3A4TSHR
SCHEMBL29181814 0.68 IDO1 (0.44) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL27945532 0.68 IDO1 (0.44) IDO1EP300KAT8ALDH1A1GAA
SCHEMBL23515356 0.67 IDO1 (0.51) IDO1EP300KAT8MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965147-B Benzofuran derivatives 武田药品工业株式会社 2016-08-24 CN disclosed