SCHEMBL28076832

SCHEMBL28076832

Cc1cc(-c2ccc(N(C)C)cc2)c2c(c1C)OC(C)(C)C2=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
PGR P06401 4/20 0.36
GPR84 Q9NQS5 1/20 0.36
ALDH1A1 P00352 3/20 0.35
HPGD P15428 2/20 0.35
CYP3A4 P08684 1/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B10 Q99714 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ACHE P22303 1/20 0.32
TNKS O95271 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NOTUM Q6P988 1/20 0.32
HTR6 P50406 1/20 0.32
APP P05067 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL659388 0.77 MAPT (0.36) MAPTPGRALDH1A1HPGDCYP3A4
SCHEMBL659098 0.74 KDM4E (0.31) ALDH1A1HPGD
SCHEMBL8719849 0.65 ALDH1A1 (0.43) MAPTPGRALDH1A1HPGDCYP3A4
SCHEMBL659806 0.65 ESR1 (0.42) ALDH1A1HPGDTDP1
SCHEMBL3600806 0.64 NQO1 (0.33) ALDH1A1HPGD
SCHEMBL24625462 0.63 ALDH1A1 (0.50) MAPTPGRALDH1A1HPGDCYP3A4
SCHEMBL9052702 0.63 MEN1 (0.50) MAPTPGRALDH1A1HPGDCYP3A4
SCHEMBL10795565 0.62 ALDH1A1 (0.52) MAPTPGRALDH1A1CYP3A4HSD17B10
SCHEMBL3603579 0.61 TSHR (0.31) ALDH1A1
SCHEMBL8712948 0.61 MAPT (0.35) MAPTALDH1A1HSD17B10CRHBPCRHR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965147-B Benzofuran derivatives 武田药品工业株式会社 2016-08-24 CN disclosed