SCHEMBL28077284

SCHEMBL28077284

Nc1ccc(S(N)(=O)=O)c(-c2ccc3c(c2)CNCC3)c1

nearest known ligand 0.57

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PNMT P11086 9/20 0.55
ADRA2A P08913 2/20 0.55
ADRA2B P18089 2/20 0.55
ADRA2C P18825 2/20 0.55
CD274 Q9NZQ7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14362208 0.84 PNMT (0.57) PNMTADRA2AADRA2BADRA2CCD274
SCHEMBL29521679 0.75 PNMT (0.60) PNMTADRA2AADRA2BADRA2C
SCHEMBL330080 0.75 PNMT (0.60) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL3285222 0.74 PNMT (0.58) PNMTADRA2AADRA2BADRA2C
SCHEMBL671916 0.74 CA1 (0.50)
Hydrochloric Acid SCHEMBL4517857 0.74 PNMT (0.58) PNMTADRA2AADRA2BADRA2C
SCHEMBL29941551 0.71 PNMT (1.00) PNMTADRA2AADRA2BADRA2C
SCHEMBL1487047 0.71 PNMT (1.00) PNMTADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL1038022 0.70 PNMT (0.97) PNMTADRA2AADRA2BADRA2C
SCHEMBL7207915 0.69 PNMT (0.50) PNMTADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105764510-A An H3 receptor antagonist combined with a cholinesterase inhibitor for use in the treatment of alzheimer's disease 赛诺菲 2016-07-13 CN disclosed