SCHEMBL28077549

SCHEMBL28077549

O=C(O)N1CCC(CO)(c2ccc(C(F)F)cc2)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 3/20 0.43
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
PKLR P30613 1/20 0.34
PRKAB2 O43741 5/20 0.33
PRKAG1 P54619 5/20 0.33
PRKAA2 P54646 5/20 0.33
PRKAA1 Q13131 5/20 0.33
PRKAG3 Q9UGI9 5/20 0.33
PRKAG2 Q9UGJ0 5/20 0.33
PRKAB1 Q9Y478 5/20 0.33
TACR1 P25103 2/20 0.33
CCR1 P32246 1/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 2/20 0.32
USP2 O75604 1/20 0.32
GRM2 Q14416 1/20 0.32
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2425390 0.84 HSD11B1 (0.49) HSD11B1DRD2DRD4DRD3
SCHEMBL2425376 0.82 HSD11B1 (0.58) HSD11B1PKLRTACR1CCR1CYP2D6
SCHEMBL16554013 0.81 TACR1 (0.48) HSD11B1TACR1USP2
SCHEMBL21078011 0.81 JAK2 (0.34) HSD11B1JAK2JAK1CCR1DRD2
SCHEMBL3585852 0.81 HSD11B1 (0.45) HSD11B1PKLRTACR1CCR1
SCHEMBL16565155 0.81 JAK2 (0.41) HSD11B1JAK2JAK1TACR1CCR1
SCHEMBL28123227 0.80 TACR1 (0.44) HSD11B1TACR1
SCHEMBL16554014 0.78 JAK2 (0.33) HSD11B1JAK2JAK1
SCHEMBL3589814 0.78 HSD11B1 (0.45) HSD11B1PKLRTACR1CYP3A4CYP2D6
SCHEMBL28077736 0.77 HSD11B1 (0.43) HSD11B1JAK2JAK1PRKAB2PRKAG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745209-A Triazolopyridine compounds, compositions, and methods of use thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed