SCHEMBL28078253

SCHEMBL28078253

NC(CCCc1ccccn1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.55
CYP2C19 P33261 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PTPRA P18433 1/20 0.51
SLC1A5 Q15758 1/20 0.51
HRH1 P35367 2/20 0.50
NOS1 P29475 3/20 0.49
GRIK1 P39086 1/20 0.47
POLB P06746 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45
ARG1 P05089 1/20 0.44
KIF11 P52732 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28078250 1.00 CYP1A2 (0.55) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL28102642 0.94 HRH1 (0.55) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL28102643 0.94 HRH1 (0.55) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL30428132 0.90 SLC1A5 (0.56) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL1768948 0.90 SLC1A5 (0.56) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL1176394 0.90 SLC1A5 (0.56) CYP1A2CYP2C19SMN1; SMN2PTPRASLC1A5
SCHEMBL27734507 0.88 CYP1A2 (0.51) CYP1A2CYP2C19SMN1; SMN2PTPRAHRH1
SCHEMBL27734504 0.88 CYP1A2 (0.51) CYP1A2CYP2C19SMN1; SMN2PTPRAHRH1
Ornithine Aketoglutarate SCHEMBL3838101 0.82 PTPRA (0.54) CYP1A2PTPRASLC1A5HRH1GRIN2D
Ornithine SCHEMBL3838093 0.82 PTPRA (0.54) CYP1A2PTPRASLC1A5HRH1GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107636007-A Beta hairpin peptide mimics 波利弗尔股份公司 2018-01-26 CN disclosed
CN-107001426-A Beta-hairpin peptidomimetics 波利弗尔股份公司 2017-08-01 CN disclosed
CN-107001425-A Beta hairpin peptide mimics 波利弗尔股份公司 2017-08-01 CN disclosed
CN-102844327-B Template-fixed peptidomimetics with CXCR7 modulatory activity 波利弗尔股份公司 2016-10-26 CN disclosed
CN-105849119-A Beta-hairpin peptidomimetics 波利弗尔股份公司 2016-08-10 CN disclosed
CN-105324390-A Beta-hairpin peptidomimetics POLYPHOR AG 2016-02-10 CN disclosed