SCHEMBL28078557

SCHEMBL28078557

COc1ccc(-n2cc(-c3ccccc3C)c(C(=O)O)c2C(F)(F)F)cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 2/20 0.43
PDE5A O76074 1/20 0.41
KCNH2 Q12809 1/20 0.41
GRM1 Q13255 1/20 0.41
GFER P55789 1/20 0.41
PTPN11 Q06124 2/20 0.41
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
NPSR1 Q6W5P4 1/20 0.39
PPARG P37231 1/20 0.38
ABCG2 Q9UNQ0 2/20 0.38
PTGS2 P35354 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
PDE11A Q9HCR9 1/20 0.37
RPA1 P27694 1/20 0.37
PTGS1 P23219 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28078365 0.91 PDE5A (0.40) CMA1PDE5AKCNH2GRM1GFER
SCHEMBL28078523 0.89 PDE5A (0.39) CMA1PDE5AKCNH2GRM1GFER
SCHEMBL28078543 0.89 KDM4E (0.45) KDM4EMAPTNPSR1ABCG2ALDH1A1
SCHEMBL28078423 0.88 PTGS2 (0.40) MAPTABCG2PTGS2PTGS1
SCHEMBL28078534 0.86 CNR1 (0.40) KDM4EMAPTPTGS2ALDH1A1HPGD
SCHEMBL28078364 0.82 ATM (0.40) ABCG2PTGS2ALDH1A1TP53
SCHEMBL28078505 0.81 GFER (0.50) GFERPTPN11KDM4EMAPTALDH1A1
SCHEMBL28078528 0.81 JAK1 (0.36) MAPTPTGS2ALDH1A1HPGDPTGS1
SCHEMBL28078369 0.81 RPA1 (0.39) MAPTALDH1A1RPA1
SCHEMBL28078548 0.79 ABCB1 (0.37) MAPTABCG2PTGS2PDE11APTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646322-A Perfluoroalkyl pyrrole derivative and synthesis method thereof 上海大学 2016-06-08 CN disclosed