SCHEMBL28079385

SCHEMBL28079385

CCNc1cnn(-c2cccc(Br)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
RXRA P19793 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
CACNA2D1 P54289 1/20 0.39
EGFR P00533 1/20 0.38
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MAPK8 P45983 3/20 0.35
MAPK10 P53779 3/20 0.35
DRD4 P21917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28079216 0.84 PTGDR2 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL20729400 0.83 NPC1 (0.44) MKNK1RXRAGRIN1GRIN2BMAPK8
SCHEMBL28079268 0.79 DDB1 (0.43) MKNK1PTGDR2RXRAGRIN1GRIN2B
SCHEMBL2690290 0.77 CYP2A6 (0.45) MKNK1
SCHEMBL28192194 0.75 ALDH1A1 (0.50) PTGDR2ALDH1A1SMN1; SMN2MAPK8MAPK10
SCHEMBL31517551 0.72 PTGDR2 (0.46) PTGDR2RXRAGRIN1GRIN2BMEN1
SCHEMBL31517384 0.72 PTGDR2 (0.43) PTGDR2RXRAGRIN1GRIN2BMEN1
SCHEMBL1419332 0.70 EGFR (0.56) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL20560807 0.70 MEN1 (0.46) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL13835994 0.70 PTGDR2 (0.55) PTGDR2MEN1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105658640-A Alkynyl alcohols and methods of use 豪夫迈·罗氏有限公司 2016-06-08 CN disclosed