SCHEMBL28081599

SCHEMBL28081599

CCCCOc1ncc2cc[nH]c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.39
CYP3A4 P08684 6/20 0.39
CYP2C9 P11712 6/20 0.39
CYP2C19 P33261 5/20 0.39
CYP19A1 P11511 4/20 0.39
CYP1A2 P05177 3/20 0.39
FGFR1 P11362 2/20 0.35
KDR P35968 2/20 0.35
CDK1 P06493 2/20 0.35
CDK2 P24941 2/20 0.35
MAPK1 P28482 2/20 0.35
AXL P30530 2/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
CHUK O15111 1/20 0.35
PDPK1 O15530 1/20 0.35
DYRK3 O43781 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29944813 0.83 FGFR1 (0.35) FGFR1KDRMAPK1AXLCDK8
SCHEMBL12986192 0.79 FGFR1 (0.36) CYP3A4CYP1A2FGFR1KDRMAPK1
SCHEMBL1093257 0.78 BRD4 (0.43) CYP1A2FGFR1KDRMAPK1AXL
SCHEMBL1763317 0.77 GPR84 (0.38) FGFR1KDRAXLRAB9ASMN1; SMN2
SCHEMBL13021084 0.75 CYP1A2 (0.40) CYP2D6CYP3A4CYP2C9CYP2C19CYP19A1
SCHEMBL5067972 0.74 AXL (0.38) FGFR1KDRCDK1CDK2MAPK1
SCHEMBL21462266 0.74 TLR7 (0.42) CYP2D6CYP3A4TTBK1TTBK2
SCHEMBL1444090 0.71 MEN1 (0.46) CDK2RAB9ASMN1; SMN2HPGDLMNA
SCHEMBL16266763 0.69 MERTK (0.37) FGFR1KDRAXLCDC7CHEK1
SCHEMBL20508764 0.69 DYRK1A (0.38) FGFR1KDRPIM1DYRK1AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105906631-A Compounds and methods for kinase modulation, and indications therefor 普莱希科公司 2016-08-31 CN disclosed