SCHEMBL28083408

SCHEMBL28083408

O=C(O)C1(c2c(Cl)ccc(F)c2Cl)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.50
AKR1C2 P52895 5/20 0.50
APP P05067 5/20 0.50
CYP2C19 P33261 4/20 0.50
CYP3A4 P08684 4/20 0.50
CYP2C9 P11712 3/20 0.50
PSEN1 P49768 1/20 0.50
PSEN2 P49810 1/20 0.50
APH1B Q8WW43 1/20 0.50
NCSTN Q92542 1/20 0.50
APH1A Q96BI3 1/20 0.50
PSENEN Q9NZ42 1/20 0.50
AKR1C1 Q04828 4/20 0.49
HDAC4 P56524 1/20 0.41
CYP2D6 P10635 1/20 0.39
AKR1B10 O60218 1/20 0.38
AKR1C4 P17516 1/20 0.38
USP2 O75604 1/20 0.36
HTT P42858 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28083366 0.88 HDAC4 (0.42) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL20242254 0.81 HDAC4 (0.60) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL31294736 0.77 AKR1C1 (0.45) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL20242053 0.77 AKR1C3 (0.45) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL31759482 0.77 AKR1C3 (0.53) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL3373867 0.75 HDAC4 (0.70) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL9314481 0.74 AKR1C1 (0.45) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL4813224 0.73 HDAC4 (0.68) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL31759329 0.72 APP (0.69) AKR1C3AKR1C2APPCYP2C19CYP3A4
SCHEMBL2794766 0.72 AKR1C3 (0.64) AKR1C3AKR1C2APPCYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105712992-A Compound serving as cMet inhibitor and preparation method and application of compound 上海科州药物研发有限公司 2016-06-29 CN disclosed