SCHEMBL28085655

SCHEMBL28085655

COc1ccc(-c2c(COc3ccc(N)c(O)c3)c3ccccc3oc2=O)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.58
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
NPC1 O15118 3/20 0.47
VKORC1 Q9BQB6 2/20 0.47
CYP19A1 P11511 1/20 0.46
KDM4E B2RXH2 5/20 0.45
ALDH1A1 P00352 5/20 0.45
MAPT P10636 3/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HTT P42858 1/20 0.45
HPGD P15428 2/20 0.45
GAA P10253 1/20 0.45
ALOX15 P16050 1/20 0.45
ESR1 P03372 1/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085539 0.78 CYP19A1 (0.59) MAOBNPC1CYP19A1KDM4EALDH1A1
SCHEMBL31511411 0.78 MAOB (0.67) MAOBCA1CA2NPC1VKORC1
SCHEMBL11485562 0.75 MAOB (1.00) MAOBCA1CA2NPC1VKORC1
SCHEMBL8934551 0.72 VKORC1 (0.66) MAOBCA1CA2VKORC1CYP19A1
SCHEMBL28085675 0.72 MAOB (0.65) MAOBNPC1CYP19A1KDM4EALDH1A1
SCHEMBL5557246 0.71 NPC1 (0.72) MAOBNPC1CYP19A1KDM4EALDH1A1
SCHEMBL7117054 0.71 MAOB (0.72) MAOBCA1CA2NPC1VKORC1
SCHEMBL31511409 0.71 MAOB (0.72) MAOBCA1CA2NPC1VKORC1
SCHEMBL7463411 0.71 MAOB (0.72) MAOBCA1CA2NPC1VKORC1
SCHEMBL28143005 0.71 MAOB (0.72) MAOBCA1CA2NPC1VKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed