SCHEMBL11485562

SCHEMBL11485562

COc1ccc(-c2c(O)c3ccccc3oc2=O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 1.00
KDM4E B2RXH2 4/20 0.63
ALDH1A1 P00352 3/20 0.63
CYP3A4 P08684 2/20 0.63
HSD17B10 Q99714 2/20 0.63
VKORC1 Q9BQB6 2/20 0.62
NQO1 P15559 1/20 0.62
MAPT P10636 3/20 0.60
POLB P06746 2/20 0.60
TP53 P04637 2/20 0.60
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
MEN1 O00255 1/20 0.59
KMT2A Q03164 1/20 0.59
HPGD P15428 2/20 0.58
TDP1 Q9NUW8 1/20 0.58
GAA P10253 1/20 0.58
ALOX15 P16050 1/20 0.58
NPC1 O15118 2/20 0.55
ABCG2 Q9UNQ0 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5426832 0.86 MAOB (0.75) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL7117054 0.84 MAOB (0.72) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL28143005 0.84 MAOB (0.72) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL31511409 0.84 MAOB (0.72) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL7463411 0.84 MAOB (0.72) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL27790298 0.84 MAOB (0.72) MAOBKDM4EALDH1A1CYP3A4NQO1
SCHEMBL5141444 0.83 MAOB (0.71) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL11479069 0.83 MAOB (0.71) MAOBKDM4EALDH1A1CYP3A4HSD17B10
SCHEMBL669375 0.83 MAOB (0.70) MAOBKDM4EALDH1A1CYP3A4VKORC1
SCHEMBL29466790 0.83 MAOB (0.70) MAOBKDM4EALDH1A1CYP3A4VKORC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801544-A 3-aryl-4-arylamine-coumarin derivative and preparing method and medical application thereof 中国药科大学 2016-07-27 CN disclosed
US-4230850-A HYPOTENSIVE AGENTS, VASODILATION LIPHA, LYONNAISE INDUSTRIELLE PHARMACEUTIQUE (FR) 1980-10-28 US disclosed