SCHEMBL28085703

SCHEMBL28085703

C=CCOCCSc1cccc(Nc2nc(Cl)ncc2Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 3/20 0.40
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
EGFR P00533 7/20 0.39
CTSC P53634 7/20 0.39
BTK Q06187 4/20 0.38
BCL6 P41182 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28085704 0.83 CCNA2 (0.38) EGFR
SCHEMBL1025353 0.81 BCL6 (0.41) JAK3JAK2JAK1EGFRCTSC
SCHEMBL1024220 0.79 ALK (0.40) JAK3JAK2JAK1EGFRCTSC
SCHEMBL1026332 0.79 BCL6 (0.41) JAK3JAK2JAK1EGFRCTSC
SCHEMBL1027094 0.77 BCL6 (0.43) JAK3JAK2JAK1EGFRCTSC
SCHEMBL28085696 0.75 JAK3 (0.39) JAK3JAK2JAK1EGFRCTSC
SCHEMBL1025568 0.75 CTSC (0.42) JAK3EGFRCTSCBTK
SCHEMBL13669984 0.74 CTSC (0.39) JAK3JAK2JAK1EGFRCTSC
SCHEMBL1025065 0.74 PIN1 (0.43) EGFR
SCHEMBL1026960 0.73 EGFR (0.37) JAK3JAK2JAK1EGFRCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105801603-A ALK inhibitor with macrocyclic structure and preparation method thereof 成都倍特药业有限公司 2016-07-27 CN disclosed