Eprazinone

Eprazinone

SCHEMBL28086279

CCOC(CN1CCN(CC(C)C(=O)c2ccccc2)CC1)c1ccccc1.N[C@@H](CSCC(=O)O)C(=O)O

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 7/20 0.46
ALDH1A1 P00352 6/20 0.46
MC4R P32245 5/20 0.42
MC1R Q01726 1/20 0.40
SMN1; SMN2 Q16637 7/20 0.39
PAX8 Q06710 2/20 0.39
JAK2 O60674 2/20 0.39
MITF O75030 4/20 0.38
HTT P42858 2/20 0.38
RAB9A P51151 2/20 0.38
GFER P55789 1/20 0.38
ATM Q13315 1/20 0.38
CHRM2 P08172 2/20 0.37
ADRA2B P18089 2/20 0.37
DRD3 P35462 2/20 0.37
SIGMAR1 Q99720 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
CYP2D6 P10635 1/20 0.37
ADRA2C P18825 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Eprazinone SCHEMBL20156 0.85 ALDH1A1 (0.57) LMNAALDH1A1MC4RMC1RSMN1; SMN2
Eprazinone SCHEMBL21807703 0.84 ALDH1A1 (0.60) LMNAALDH1A1MC4RMC1RSMN1; SMN2
Eprazinone SCHEMBL598430 0.84 ALDH1A1 (0.60) LMNAALDH1A1MC4RMC1RSMN1; SMN2
Eprazinone SCHEMBL6429748 0.84 ALDH1A1 (0.56) LMNAALDH1A1MC4RMC1RSMN1; SMN2
Eprazinone SCHEMBL1009370 0.77 ALDH1A1 (0.39) LMNAALDH1A1MC4RMC1RSMN1; SMN2
Eprazinone SCHEMBL28086760 0.74 ALDH1A1 (0.45) LMNAALDH1A1MC4RMC1RSMN1; SMN2
SCHEMBL12847710 0.67 GAA (0.58) ALDH1A1MC4RCHRM2DRD3CYP2D6
SCHEMBL14791780 0.67 POLB (0.47) LMNAALDH1A1SMN1; SMN2PAX8MITF
SCHEMBL9170851 0.67 ALDH1A1 (0.73) LMNAALDH1A1MC4RMC1RSMN1; SMN2
SCHEMBL12847709 0.66 POLB (0.55) LMNAALDH1A1SMN1; SMN2PAX8JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed