Fludiazepam

Fludiazepam

SCHEMBL28086296

CN1C(=O)CN=C(c2ccccc2F)c2cc(Cl)ccc21.O=C1CN=C(c2ccccc2)c2cc(Cl)ccc2N1

nearest known ligand 0.70

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.70
GABRA1 P14867 8/20 0.68
GABRA5 P31644 8/20 0.68
GABRA3 P34903 8/20 0.68
GABRA2 P47869 8/20 0.68
GABRB2 P47870 8/20 0.68
GABRG2 P18507 6/20 0.68
GABRB3 P28472 6/20 0.68
OPRK1 P41145 4/20 0.68
GABRP O00591 3/20 0.68
GABRD O14764 3/20 0.68
GABRB1 P18505 3/20 0.68
GABRA4 P48169 3/20 0.68
GABRE P78334 3/20 0.68
GABRA6 Q16445 3/20 0.68
GABRG1 Q8N1C3 3/20 0.68
GABRG3 Q99928 3/20 0.68
GABRQ Q9UN88 3/20 0.68
KCNH2 Q12809 2/20 0.68
CACNA1F O60840 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diazepam SCHEMBL8931438 0.93 GABRA1 (0.79) LMNAGABRA1GABRA5GABRA3GABRA2
Diazepam SCHEMBL6823824 0.93 GABRA1 (0.79) LMNAGABRA1GABRA5GABRA3GABRA2
Diazepam SCHEMBL1003950 0.91 GABRA1 (0.70) LMNAGABRA1GABRA5GABRA3GABRA2
Flunitrazepam SCHEMBL8364961 0.89 GABRA1 (0.64) LMNAGABRA1GABRA5GABRA3GABRA2
Flunitrazepam SCHEMBL28086646 0.86 GABRA1 (0.75) LMNAGABRA1GABRA5GABRA3GABRA2
Fludiazepam SCHEMBL29440251 0.86 GABRA1 (0.72) LMNAGABRA1GABRA5GABRA3GABRA2
Fludiazepam SCHEMBL29688065 0.86 GABRA1 (0.72) LMNAGABRA1GABRA5GABRA3GABRA2
Fludiazepam SCHEMBL156039 0.86 GABRA1 (0.72) LMNAGABRA1GABRA5GABRA3GABRA2
Fludiazepam SCHEMBL29564860 0.86 GABRA1 (0.72) LMNAGABRA1GABRA5GABRA3GABRA2
Fludiazepam SCHEMBL29040947 0.84 GABRA1 (0.70) LMNAGABRA1GABRA5GABRA3GABRA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103717597-B Heterocyclic compounds as kinase inhibitors 原真股份有限公司 2017-07-04 CN disclosed
CN-103492389-B Pyrazolo [4,3-d] pyrimidine as inhibitors of kinases 原真股份有限公司 2016-09-14 CN disclosed