SCHEMBL28086653

SCHEMBL28086653

COc1cccc2sc(C=O)cc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.55
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54
SLC9A1 P19634 2/20 0.49
CYP2A6 P11509 2/20 0.47
MAPK1 P28482 2/20 0.42
MAPK3 P27361 1/20 0.42
MAP2K1 Q02750 1/20 0.42
ERN1 O75460 2/20 0.41
TLR2 O60603 1/20 0.41
TLR1 Q15399 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10076720 0.79 CYP2A6 (0.42) CA2CYP2A6ERN1NPC1RAB9A
SCHEMBL4803355 0.77 CA2 (0.55) CA2HDAC3HDAC4HDAC1HDAC7
SCHEMBL5153435 0.76 NPC1 (0.50) HDAC4HDAC2HDAC8SLC9A1CYP2A6
SCHEMBL24447297 0.75 CA2 (0.57) CA2HDAC3HDAC4HDAC1HDAC7
SCHEMBL12095346 0.75 CYP2A6 (0.53) SLC9A1CYP2A6ERN1ALDH1A1L3MBTL1
SCHEMBL28020760 0.75 CA2 (0.57) CA2HDAC3HDAC4HDAC1HDAC7
SCHEMBL12095302 0.74 CYP2A6 (0.52) CA2HDAC3HDAC4HDAC1HDAC7
SCHEMBL12095282 0.74 CYP2A6 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4861203 0.74 CYP2A6 (0.52) CA2SLC9A1CYP2A6ALDH1A1ALOX15
SCHEMBL2173724 0.74 CA2 (0.59) CA2HDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103992310-B One group replaces benzo heterocyclic amine derivant and preparation method thereof and the related application as IMPDH inhibitor 中国医学科学院医药生物技术研究所 2016-07-06 CN disclosed