SCHEMBL28089940

SCHEMBL28089940

O=C(O)c1cnc2cnc[nH]c1-2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.39
ALDH1A1 P00352 2/20 0.39
TSHR P16473 2/20 0.39
GABRA1 P14867 2/20 0.39
GABRA5 P31644 2/20 0.39
GABRB2 P47870 2/20 0.39
GABRA4 P48169 2/20 0.39
NFKB1 P19838 1/20 0.39
GABRR1 P24046 1/20 0.39
GABRR2 P28476 1/20 0.39
KDM4E B2RXH2 3/20 0.38
MAPT P10636 1/20 0.38
PMP22 Q01453 1/20 0.38
KDM6B O15054 1/20 0.38
KDM4A O75164 1/20 0.38
KDM4D Q6B0I6 1/20 0.38
HIF1AN Q9NWT6 1/20 0.38
KDM2A Q9Y2K7 1/20 0.38
BLM P54132 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14250023 0.84 PARP1 (0.37) CYP3A4ALDH1A1TSHRGABRA1GABRA5
Hydrochloric Acid SCHEMBL1439124 0.82 PARP1 (0.36) CYP3A4ALDH1A1TSHRGABRA1GABRA5
SCHEMBL14949552 0.81 NPC1 (0.36) CYP3A4ALDH1A1TSHRGABRA1GABRA5
SCHEMBL3613510 0.72 IDO1 (0.42) CYP3A4ALDH1A1KDM4EPMP22NPSR1
SCHEMBL21713005 0.70 CYP3A4 (0.39) CYP3A4ALDH1A1TSHRGABRA1GABRA5
SCHEMBL798220 0.68 NAPRT (0.45) CYP3A4ALDH1A1TSHRGABRA1GABRA5
SCHEMBL4067921 0.68 ALDH1A1 (0.34) CYP3A4ALDH1A1IDO1SMN1; SMN2
SCHEMBL1402162 0.68 IDO1 (0.41) CYP3A4ALDH1A1TSHRMAPTNPSR1
SCHEMBL13725534 0.68 KMT2A (0.33) CYP3A4ALDH1A1TSHRKDM4EBLM
4-Imidazolecarboxylic Acid SCHEMBL28085192 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4238967-A1 ARYLAMIDE COMPOUND, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD THEREFOR AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2023-09-06 EP disclosed
CN-103582644-B Phthalazinone-Pyrrolopyrimidine Carboxamide Derivatives 塔科达有限责任公司 2016-07-20 CN disclosed