SCHEMBL28090568

SCHEMBL28090568

CC(C)(C)OC(N)=O.O=C(c1ccccc1)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.55
MAPT P10636 5/20 0.54
TP53 P04637 1/20 0.52
ALDH1A1 P00352 6/20 0.51
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
POLB P06746 2/20 0.49
CTDSP1 Q9GZU7 1/20 0.49
PRSS1 P07477 1/20 0.49
PRSS2 P07478 1/20 0.49
PRSS3 P35030 1/20 0.49
NPC1 O15118 3/20 0.47
RAB9A P51151 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
HPGD P15428 1/20 0.47
CCNA2 P20248 1/20 0.47
CDK2 P24941 1/20 0.47
HTT P42858 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28090586 0.88 MAPK1 (0.57) TSHRMAPTALDH1A1CES2CES1
Dinitrophenylene SCHEMBL28255199 0.86 TSHR (0.55) TSHRMAPTTP53ALDH1A1CES2
SCHEMBL27384308 0.85 MAPT (0.50) TSHRMAPTTP53ALDH1A1CES2
SCHEMBL27406857 0.85 MAPT (0.61) TSHRMAPTTP53ALDH1A1CES2
Carbamic Acid SCHEMBL27919491 0.85 TSHR (0.70) TSHRMAPTTP53ALDH1A1CES2
Chloromethane SCHEMBL27475705 0.85 TP53 (0.67) TSHRMAPTTP53ALDH1A1CES2
Nitrobenzene SCHEMBL27619171 0.85 ALDH1A1 (0.53) TSHRMAPTTP53ALDH1A1CES2
Urea SCHEMBL28125526 0.85 TSHR (0.70) TSHRMAPTTP53ALDH1A1CES2
Methylamine SCHEMBL27764628 0.85 TP53 (0.67) TSHRMAPTTP53ALDH1A1CES2
Hydrazine SCHEMBL27600958 0.83 TP53 (0.69) TSHRMAPTTP53ALDH1A1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109311813-A The functionalized universal ligand of the meta position-C-H of palladium chtalyst 斯克利普斯研究院 2019-02-05 CN disclosed
CN-108055843-A Synthesis of benzodiazepine derivatives 特里奥医药有限公司 2018-05-18 CN disclosed
CN-106715411-A Benzodiazepine derivatives as cck2/gastrin receptor antagonists 特里奥医药有限公司 2017-05-24 CN disclosed
CN-104245671-B nitrogen-containing heterocyclic compound or salt thereof 富士胶片株式会社 2017-03-22 CN disclosed
CN-106279172-A Purinone compound as inhibitors of kinases 药品循环有限责任公司 2017-01-04 CN disclosed
CN-104640861-B Purinone compounds as kinase inhibitors 药品循环公司 2016-08-24 CN disclosed