SCHEMBL28091997

SCHEMBL28091997

Nc1ncnc2[nH]nc(C3CCCNC3)c12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.36
JAK1 P23458 1/20 0.36
JAK3 P52333 1/20 0.36
BTK Q06187 1/20 0.36
METTL3 Q86U44 1/20 0.36
IKBKB O14920 1/20 0.35
ACVRL1 P37023 2/20 0.35
CHEK1 O14757 2/20 0.34
CCNA2 P20248 2/20 0.34
CDK2 P24941 2/20 0.34
CCNA1 P78396 2/20 0.34
EGFR P00533 2/20 0.34
SRC P12931 2/20 0.34
RET P07949 1/20 0.34
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
PRKDC P78527 2/20 0.33
ULK1 O75385 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16075033 0.84 RET (0.38) SRCRETPIK3CDPIK3CAPIK3CB
SCHEMBL29778119 0.77 IRAK4 (0.39) JAK2JAK1RETPIK3CDPIK3CA
SCHEMBL30515860 0.71 EGFR (0.33) ACVRL1EGFRSRCABL1
SCHEMBL9900029 0.71 BTK (0.46) JAK2JAK1JAK3BTKIKBKB
SCHEMBL9900173 0.71 BTK (0.46) JAK2JAK1JAK3BTKIKBKB
Hydrochloric Acid SCHEMBL16654494 0.70 PIK3CD (0.53) BTKSRCPIK3CDPIK3CAPIK3CB
SCHEMBL30387689 0.69 PIK3CD (0.65) BTKPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL28063328 0.68 CHEK1 (0.42) IKBKBCHEK1CCNA2CDK2CCNA1
SCHEMBL28345670 0.68 JAK3 (0.59) JAK2JAK1JAK3
SCHEMBL1536074 0.67 JAK2 (0.52) JAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105985343-A Preparation method for ibrutinib 上海昶朗医药科技有限公司 2016-10-05 CN disclosed