SCHEMBL28097122

SCHEMBL28097122

CN(C)C1CCN(c2cncnc2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.46
CHRNB2 P17787 2/20 0.45
CHRNB4 P30926 2/20 0.45
CHRNA3 P32297 2/20 0.45
CHRNA4 P43681 2/20 0.45
L3MBTL3 Q96JM7 1/20 0.39
DPP4 P27487 1/20 0.37
DPP8 Q6V1X1 1/20 0.37
DPP9 Q86TI2 1/20 0.37
DPP7 Q9UHL4 1/20 0.37
CCNE1 P24864 1/20 0.37
CDK2 P24941 1/20 0.37
HSF1 Q00613 1/20 0.37
CHI3L1 P36222 1/20 0.36
KCNH2 Q12809 1/20 0.36
CHIT1 Q13231 1/20 0.36
CHIA Q9BZP6 1/20 0.36
OPRM1 P35372 2/20 0.36
OPRL1 P41146 2/20 0.36
MAP4K4 O95819 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20311336 0.80 ACVR1 (0.42) L3MBTL3CCNE1CDK2HSF1KCNH2
SCHEMBL22837854 0.80 NPY5R (0.53) CYP3A4CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL16892009 0.79 PTPN11 (0.42) L3MBTL3CCNE1CDK2HSF1MAP4K4
SCHEMBL19152362 0.79 CHRNB2 (0.49) CYP3A4CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL19947418 0.78 CHRNB2 (0.53) CYP3A4CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL2362576 0.78 CHKA (0.53) CYP3A4L3MBTL3
SCHEMBL25085650 0.76 ACVR1 (0.38) L3MBTL3CCNE1CDK2HSF1KCNH2
SCHEMBL21267364 0.76 CDK4 (0.40) L3MBTL3CCNE1CDK2HSF1PTPN11
SCHEMBL26149309 0.75 ACVR1 (0.41) L3MBTL3PTPN11ACVR1
SCHEMBL2266909 0.75 CHRNB2 (0.49) CYP3A4CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108779117-A Kinase inhibitor 重庆复创医药研究有限公司 2018-11-09 CN disclosed
CN-105916848-B Kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2018-01-09 CN disclosed
CN-105916848-A Kinase inhibitors and uses thereof 山东轩竹医药科技有限公司 2016-08-31 CN disclosed