SCHEMBL28097458

SCHEMBL28097458

[CH2]C[C@](C)(N)c1cc([N+](=O)[O-])ccc1F

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.46
HIF1A Q16665 1/20 0.46
HTT P42858 3/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
GAA P10253 2/20 0.44
THRB P10828 1/20 0.44
POLB P06746 2/20 0.41
KMT2A Q03164 3/20 0.40
MAPT P10636 1/20 0.40
TDP1 Q9NUW8 3/20 0.39
CYP3A4 P08684 2/20 0.39
TSHR P16473 2/20 0.38
MEN1 O00255 1/20 0.38
GALR3 O60755 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PDE7A Q13946 1/20 0.37
S1PR4 O95977 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1981365 0.87 ALDH1A1 (0.51) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL1977121 0.83 ALDH1A1 (0.45) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL12077461 0.83 ALDH1A1 (0.45) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL1977119 0.83 ALDH1A1 (0.45) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL9898944 0.82 ALDH1A1 (0.47) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL9898940 0.82 ALDH1A1 (0.47) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL4077302 0.82 ALDH1A1 (0.47) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL12350182 0.82 ALDH1A1 (0.47) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL18856053 0.82 ALDH1A1 (0.43) ALDH1A1HIF1AHTTL3MBTL1GAA
SCHEMBL13466033 0.81 ALDH1A1 (0.42) ALDH1A1HIF1AHTTL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103429590-B 1, 4 thiazepine/sulfone as BACE1 and/or BACE2 inhibitors 霍夫曼-拉罗奇有限公司 2016-10-26 CN disclosed