SCHEMBL28098004

SCHEMBL28098004

COc1cc2ncnc(-c3cccc(N)c3)c2cc1OCCN

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KIT P10721 4/20 0.58
RET P07949 2/20 0.52
KDR P35968 2/20 0.52
EGFR P00533 5/20 0.45
ENPP1 P22413 3/20 0.44
FGFR1 P11362 1/20 0.44
FLT1 P17948 1/20 0.44
FBP1 P09467 1/20 0.44
BRD4 O60885 1/20 0.43
ERBB2 P04626 1/20 0.43
ERBB4 Q15303 1/20 0.43
ATM Q13315 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5568255 0.91 KIT (0.64) KITRETKDREGFRENPP1
SCHEMBL182873 0.78 PIK3CD (0.60) KITRETENPP1
SCHEMBL6181412 0.76 EGFR (0.63) KITRETKDREGFRATM
SCHEMBL5569432 0.76 KIT (0.69) KITRETKDREGFRENPP1
SCHEMBL4782102 0.76 WHR1 (0.61) KITRETKDREGFRATM
SCHEMBL2126095 0.75 EGFR (0.61) KITKDREGFRFGFR1FLT1
SCHEMBL2125179 0.75 EGFR (0.61) KITRETKDREGFRFLT1
SCHEMBL182424 0.75 PIK3CD (0.60) KITENPP1
SCHEMBL295984 0.74 WHR1 (0.50) KITRETKDREGFR
SCHEMBL26098937 0.74 KIT (0.56) KITRETKDREGFRENPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106045980-A Quinazoline derivative and preparation method thereof 江苏开放大学 2016-10-26 CN disclosed