Azetidine

Azetidine

SCHEMBL28099548

C1CNC1.c1ccc(Cc2nncc3ccccc23)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.53
HTT P42858 2/20 0.44
NPSR1 Q6W5P4 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
SMO Q99835 4/20 0.40
CYP3A4 P08684 3/20 0.40
LMNA P02545 2/20 0.40
CYP1A2 P05177 2/20 0.40
PRNP P04156 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
HPGD P15428 1/20 0.40
HTR2C P28335 3/20 0.39
PARP1 P09874 1/20 0.39
AR P10275 1/20 0.39
KDM4E B2RXH2 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31738482 0.91 CYP19A1 (0.61) CYP19A1HTTNPSR1MEN1KMT2A
SCHEMBL7069713 0.91 CYP19A1 (0.61) CYP19A1HTTNPSR1MEN1KMT2A
SCHEMBL29481851 0.80 CYP19A1 (0.53) CYP19A1NPSR1CYP3A4LMNACYP1A2
SCHEMBL871138 0.80 CYP19A1 (0.53) CYP19A1NPSR1CYP3A4LMNACYP1A2
Hydrochloric Acid SCHEMBL6061889 0.78 CYP19A1 (0.52) CYP19A1NPSR1CYP3A4LMNACYP1A2
SCHEMBL9807642 0.77 CYP19A1 (0.54) CYP19A1MEN1KMT2ACYP3A4LMNA
SCHEMBL28873268 0.75 CYP19A1 (0.62) CYP19A1MEN1KMT2ACYP3A4LMNA
Succinic Acid SCHEMBL21385162 0.73 KDR (0.53) CYP19A1ALDH1A1MAPT
SCHEMBL12785877 0.72 GBA1 (0.46) CYP19A1KMT2ACYP3A4LMNACYP1A2
SCHEMBL28173505 0.71 SCN9A (0.54) CYP19A1HTTNPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105985320-A Benzylphthalazine compound and its preparation method and use 复旦大学 2016-10-05 CN claimed