SCHEMBL28100490

SCHEMBL28100490

CCCCCOS(=O)(=O)Cc1ccc2nc[nH]c(=O)c2c1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 7/20 0.48
IP6K3 Q96PC2 3/20 0.48
IP6K2 Q9UHH9 3/20 0.48
PARP1 P09874 7/20 0.45
CHEK1 O14757 1/20 0.42
PIM1 P11309 1/20 0.42
AKT1 P31749 1/20 0.42
FLT3 P36888 1/20 0.42
PIM3 Q86V86 1/20 0.42
SLC2A1 P11166 1/20 0.41
ACVR1 Q04771 2/20 0.40
DHFR P00374 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17080827 0.78 IP6K1 (0.55) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL8170598 0.75 IP6K1 (0.71) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL28100493 0.74 IP6K1 (0.49) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL28100544 0.69 TP53 (0.37)
SCHEMBL22042406 0.68 IP6K1 (0.61) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL874691 0.67 HPGD (0.51)
SCHEMBL27947190 0.67 IP6K1 (0.62) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL25721982 0.66 IP6K1 (0.58) IP6K1IP6K3IP6K2PARP1CHEK1
SCHEMBL7784180 0.66 HPGD (0.50)
SCHEMBL15543392 0.66 HPGD (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106132956-B Heterocyclic compound, preparation method and application thereof 中国科学院上海药物研究所 2019-12-10 CN disclosed
CN-106132956-A Heterocyclic compound, preparation method and application thereof 中国科学院上海药物研究所 2016-11-16 CN disclosed