SCHEMBL28107488

SCHEMBL28107488

CC(C)(CC(=O)O)n1cc(-c2ccnc3[nH]ccc23)cn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 5/20 0.57
AURKA O14965 4/20 0.57
INCENP Q9NQS7 1/20 0.57
TPX2 Q9ULW0 1/20 0.57
JAK2 O60674 6/20 0.56
GRM4 Q14833 1/20 0.53
JAK1 P23458 5/20 0.48
NUDT1 P36639 1/20 0.46
JAK3 P52333 3/20 0.46
IKBKB O14920 2/20 0.46
CHUK O15111 2/20 0.46
DAPK3 O43293 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
PAK4 O96013 1/20 0.46
CSF1R P07333 1/20 0.46
RET P07949 1/20 0.46
IGF1R P08069 1/20 0.46
FGFR1 P11362 1/20 0.46
PRKACA P17612 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29540487 0.91 AURKB (0.60) AURKBAURKAINCENPTPX2JAK2
SCHEMBL101177 0.91 AURKB (0.60) AURKBAURKAINCENPTPX2JAK2
Trifluoroacetic Acid SCHEMBL4094031 0.88 JAK2 (0.54) AURKBAURKAINCENPTPX2JAK2
SCHEMBL15389320 0.87 AURKB (0.52) AURKBAURKAINCENPTPX2JAK2
SCHEMBL99992 0.87 AURKA (0.52) AURKBAURKAINCENPTPX2JAK2
SCHEMBL100576 0.86 AURKB (0.62) AURKBAURKAINCENPTPX2JAK2
SCHEMBL21085376 0.85 AURKB (0.63) AURKBAURKAINCENPTPX2JAK2
SCHEMBL21320196 0.85 JAK2 (0.75) AURKBAURKAINCENPTPX2JAK2
SCHEMBL99868 0.84 AURKB (0.59) AURKBAURKAINCENPTPX2JAK2
SCHEMBL101852 0.84 AURKA (0.54) AURKBAURKAINCENPTPX2JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103254190-B Heteroaryl substituted pyrrolo-[2,3-b] pyridine and pyrrolo-[2,3-b] pyrimidine as Janus inhibitors of kinases 因塞特控股公司 2016-12-07 CN disclosed