SCHEMBL28110409

SCHEMBL28110409

COc1cccc(-c2ncc3ccccc3n2)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 10/20 0.59
CYP3A4 P08684 8/20 0.59
CYP2C9 P11712 4/20 0.59
CYP2B6 P20813 2/20 0.59
AHR P35869 2/20 0.59
NR1I3 Q14994 2/20 0.59
VDR P11473 1/20 0.59
CLK4 Q9HAZ1 5/20 0.57
DYRK1A Q13627 1/20 0.57
CYP2D6 P10635 7/20 0.56
MAPK1 P28482 5/20 0.56
CYP2C19 P33261 5/20 0.56
USP2 O75604 4/20 0.56
HSD17B10 Q99714 3/20 0.56
ALOX15 P16050 3/20 0.56
MAPT P10636 3/20 0.53
ATM Q13315 1/20 0.53
PDGFRB P09619 1/20 0.52
PDGFRA P16234 1/20 0.52
ABCB1 P08183 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31023430 1.00 CYP1A2 (0.59) CYP1A2CYP3A4CYP2C9CYP2B6AHR
SCHEMBL8775416 0.88 CYP1A2 (0.50) CYP1A2CYP3A4CYP2C9CYP2B6AHR
SCHEMBL16404354 0.83 CYP1A2 (0.62) CYP1A2CLK4MAPTABCG2LMNA
SCHEMBL8776971 0.82 PDE10A (0.48) CYP1A2CYP3A4CYP2C9CYP2B6AHR
SCHEMBL29928263 0.80 NPC1 (0.59) HSD17B10MAPTPDGFRBPDGFRATSHR
SCHEMBL27746869 0.80 NPC1 (0.61) CYP1A2MAPTPDGFRBPDGFRAABCB1
SCHEMBL31325764 0.80 NPC1 (0.59) CYP1A2CYP3A4CYP2C9CLK4CYP2D6
SCHEMBL30483555 0.80 CYP1A2 (0.58) CYP1A2NR1I3PDE10AMEN1KMT2A
SCHEMBL19981078 0.80 CYP1A2 (0.58) CYP1A2NR1I3PDE10AMEN1KMT2A
SCHEMBL23068690 0.77 CYP1A2 (0.54) CYP1A2CYP3A4CYP2C9CYP2B6AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109879820-A A kind of synthetic method of quinazolinone heterocyclic compound 扬州大学 2019-06-14 CN disclosed
CN-106008370-B A kind of synthetic method of 2- substituted quinazoline heterocyclic compounds 温州大学 2018-12-18 CN disclosed
CN-106008370-A Synthesis method for 2-substituted quinazoline heterocyclic compound 温州大学 2016-10-12 CN disclosed