SCHEMBL28111774

SCHEMBL28111774

O=C(NC1CCCCC1)c1ccc(N2CCCCC2)nn1

nearest known ligand 0.66

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.66
ALDH1A1 P00352 6/20 0.51
CYP1A2 P05177 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2C19 P33261 2/20 0.51
MEN1 O00255 1/20 0.51
CYP2C9 P11712 1/20 0.51
KMT2A Q03164 1/20 0.51
CNR2 P34972 3/20 0.50
ACKR3 P25106 1/20 0.50
PRKAA2 P54646 1/20 0.49
HPGDS O60760 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22565386 0.91 ACKR3 (0.61) HSD11B1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL24881303 0.87 HSD11B1 (0.52) HSD11B1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL22873378 0.87 HSD11B1 (0.52) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL26366853 0.87 HSD11B1 (0.52) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL26367076 0.87 HSD11B1 (0.52) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL22565385 0.84 HSD11B1 (0.49) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL22565347 0.81 PRKAA2 (0.47) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL2591980 0.80 HSD11B1 (1.00) HSD11B1ALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL24267248 0.79 PRKAA2 (0.47) HSD11B1ALDH1A1CNR2ACKR3PRKAA2
SCHEMBL28836616 0.78 SCD (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN claimed
CN-106187910-A Pyridazine class derivant and its production and use 浙江大学 2016-12-07 CN disclosed