SCHEMBL2811187

SCHEMBL2811187

FC(F)(F)c1ccc(CNc2nc(N3CCCC3)nc3c2cnn3CCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.48
ALDH1A1 P00352 1/20 0.46
CTNNB1 P35222 6/20 0.46
TCF7L2 Q9NQB0 6/20 0.46
SRC P12931 2/20 0.46
ABL1 P00519 1/20 0.46
USP2 O75604 1/20 0.45
RAB9A P51151 1/20 0.45
PDE5A O76074 2/20 0.45
HRH4 Q9H3N8 1/20 0.45
APP P05067 1/20 0.43
ACHE P22303 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
HTR2A P28223 1/20 0.42
DRD3 P35462 1/20 0.42
PDE9A O76083 1/20 0.42
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2875828 0.90 SRC (0.52) ALDH1A1CTNNB1TCF7L2SRCABL1
SCHEMBL2786942 0.83 HRH4 (0.54) ALDH1A1SRCABL1PDE5AHRH4
SCHEMBL2835632 0.81 BCDIN3D (0.52) PDE2AALDH1A1CTNNB1TCF7L2SRC
SCHEMBL2810687 0.80 PIK3CA (0.54) ALDH1A1SRCABL1USP2RAB9A
SCHEMBL3640038 0.79 APP (0.64) ALDH1A1CTNNB1TCF7L2PDE5AHRH4
SCHEMBL3644324 0.78 CTNNB1 (0.64) ALDH1A1CTNNB1TCF7L2PDE5AHRH4
SCHEMBL3644693 0.78 HTR2C (0.58) PDE2APDE5AHRH4PDE4APDE4B
SCHEMBL2814606 0.75 CDK1 (0.42) PDE2AALDH1A1
SCHEMBL2871542 0.74 PDE5A (0.51) ALDH1A1SRCABL1USP2RAB9A
SCHEMBL2807943 0.73 SRC (0.68) SRCABL1USP2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118367-A2 ANTIVIRAL PYRIMIDINES PROGENICS PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed