SCHEMBL28111956

SCHEMBL28111956

COCOc1cccc(N)c1C

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.48
CYP3A4 P08684 1/20 0.48
PIK3CA P42336 1/20 0.48
PTPN1 P18031 1/20 0.45
ALDH1A1 P00352 4/20 0.42
TDP1 Q9NUW8 2/20 0.42
ADRA2B P18089 1/20 0.42
PTGS1 P23219 1/20 0.42
MAPT P10636 4/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
MAPK1 P28482 1/20 0.40
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
GAA P10253 2/20 0.36
HTR1B P28222 1/20 0.36
CD44 P16070 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
KDM4E B2RXH2 1/20 0.34
KCNN4 O15554 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21694155 0.85 ALDH1A1 (0.57) TSHRCYP3A4PIK3CAALDH1A1TDP1
SCHEMBL11204587 0.82 ALDH1A1 (0.63) TSHRCYP3A4PTPN1ALDH1A1TDP1
SCHEMBL21694161 0.80 CD44 (0.48) TSHRCYP3A4PIK3CAPTPN1ALDH1A1
SCHEMBL22182755 0.80 HTR1B (0.55) TSHRPTPN1ALDH1A1TDP1MAPT
SCHEMBL19400221 0.80 MAPK1 (0.47) TSHRCYP3A4PTPN1ALDH1A1TDP1
SCHEMBL1141313 0.80 ALDH1A1 (0.67) TSHRCYP3A4PIK3CAALDH1A1TDP1
SCHEMBL29617909 0.79 PTPN1 (0.42) PTPN1ALDH1A1TDP1ADRA2BPTGS1
SCHEMBL24596979 0.79 ALDH1A1 (0.41) TSHRCYP3A4PIK3CAPTPN1ALDH1A1
SCHEMBL3081933 0.79 ALDH1A1 (0.41) TSHRCYP3A4PTPN1ALDH1A1TDP1
SCHEMBL363904 0.79 ALDH1A1 (0.41) TSHRCYP3A4PIK3CAPTPN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106045923-A Histone deacetylase inhibitor and preparation method and application thereof 广东众生药业股份有限公司 2016-10-26 CN disclosed