SCHEMBL28112247

SCHEMBL28112247

O=C(OC1CCCCC1)C(F)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.41
EPHX1 P07099 2/20 0.40
NAAA Q02083 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
CYP2C19 P33261 2/20 0.36
GPR35 Q9HC97 2/20 0.35
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA9 Q16790 2/20 0.35
HTT P42858 2/20 0.34
TSHR P16473 2/20 0.33
CASP1 P29466 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MMP1 P03956 1/20 0.32
MMP9 P14780 1/20 0.32
MMP12 P39900 1/20 0.32
HDAC4 P56524 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12704999 0.79 EPHX1 (0.45) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL12705000 0.79 EPHX1 (0.45) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL11991797 0.79 EPHX1 (0.45) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL11991795 0.77 CYP19A1 (0.42) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL29163208 0.76 CYP19A1 (0.42) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL17281530 0.76 CYP19A1 (0.50) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL21396853 0.75 L3MBTL1 (0.38) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL14422659 0.74 EPHX1 (0.48) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL5008329 0.74 L3MBTL1 (0.37) CYP19A1EPHX1NAAAL3MBTL1CYP2C19
SCHEMBL5012428 0.74 L3MBTL1 (0.37) CYP19A1EPHX1NAAAL3MBTL1CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106278887-A A kind of synthetic method of 2,3,3,3 tetrafluoro propionic esters 赵满良 2017-01-04 CN disclosed