SCHEMBL28112757

SCHEMBL28112757

CC(=O)Oc1cccc2[nH]c3c(c(=O)c12)CCCC3

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
GBA1 P04062 1/20 0.41
PARP1 P09874 2/20 0.40
HSD17B10 Q99714 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 3/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
APEX1 P27695 1/20 0.39
RECQL P46063 1/20 0.39
BLM P54132 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.38
LIMK2 P53671 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28113325 0.82 KDM4E (0.38) KDM4EALDH1A1PARP1HSD17B10MAPT
SCHEMBL28113320 0.80 GBA1 (0.46) KDM4EALDH1A1SMN1; SMN2GBA1PARP1
SCHEMBL15067435 0.77 KDM4E (0.52) KDM4EALDH1A1SMN1; SMN2HSD17B10TP53
SCHEMBL28235800 0.74 ABCG2 (0.68) KDM4EALDH1A1SMN1; SMN2HSD17B10MAPT
SCHEMBL28640309 0.73 ABCG2 (0.67) KDM4EALDH1A1SMN1; SMN2HSD17B10MAPT
SCHEMBL28145530 0.73 ABCG2 (0.67) KDM4EALDH1A1SMN1; SMN2HSD17B10MAPT
SCHEMBL15069471 0.73 GFER (0.52) KDM4EALDH1A1SMN1; SMN2PARP1HSD17B10
SCHEMBL4101907 0.72 HTR2C (0.54) KDM4EALDH1A1SMN1; SMN2PARP1HSD17B10
SCHEMBL2486768 0.69 KDM4E (0.49) KDM4EALDH1A1SMN1; SMN2HSD17B10TP53
SCHEMBL6628829 0.69 HTR2C (0.54) KDM4EALDH1A1PARP1HSD17B10TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106083849-A The quaternary condensed or five-membered ring pyrido phthalazone compounds as PARP inhibitor 百济神州有限公司 2016-11-09 CN disclosed