SCHEMBL28114554

SCHEMBL28114554

Cc1cc(C(N)=O)cc(C)c1OB(O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.42
HTT P42858 2/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
PARP1 P09874 3/20 0.38
LMNA P02545 1/20 0.37
BRD4 O60885 1/20 0.36
BRD9 Q9H8M2 1/20 0.36
PARP10 Q53GL7 4/20 0.35
PARP4 Q9UKK3 2/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
PARP2 Q9UGN5 1/20 0.35
NCOA1 Q15788 1/20 0.35
NCOA3 Q9Y6Q9 1/20 0.35
BPTF Q12830 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
CYP3A4 P08684 1/20 0.34
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005872 0.79 TSHR (0.55) TSHRHTTAPOBEC3AAPOBEC3GPARP1
SCHEMBL13847870 0.78 TSHR (0.43) TSHRHTTAPOBEC3AAPOBEC3GPARP1
SCHEMBL18471225 0.73 SMN1; SMN2 (0.49) TSHRHTTAPOBEC3AAPOBEC3GPARP1
SCHEMBL10831613 0.73 PARP1 (0.46) TSHRHTTAPOBEC3AAPOBEC3GPARP1
SCHEMBL4859546 0.73 RAPGEF4 (0.36) LMNACA1CA2ALDH1A1KMT2A
SCHEMBL4687491 0.72 TSHR (0.46) TSHRHTTLMNABRD4NCOA1
SCHEMBL15492298 0.72 TSHR (0.47) TSHRHTTAPOBEC3AAPOBEC3GPARP1
SCHEMBL3220166 0.72 CA1 (0.48) TSHRPARP1LMNABRD4CA1
SCHEMBL8173238 0.72 CYP3A4 (0.44) CA1CA2SMN1; SMN2CYP3A4ALDH1A1
SCHEMBL1004660 0.72 PARP1 (0.50) TSHRHTTAPOBEC3AAPOBEC3GPARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104109115-B Phenylpropionic acid compound, its pharmaceutical composition, preparation method and the purposes of a kind of nitrogen heterocyclic ring link 中国科学院上海药物研究所 2016-11-23 CN disclosed