SCHEMBL28114780

SCHEMBL28114780

CCCCCc1ccc(Cl)c(F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.48
SIGMAR1 Q99720 2/20 0.46
RARB P10826 2/20 0.44
RARA P10276 1/20 0.44
RARG P13631 1/20 0.44
ESR1 P03372 2/20 0.44
ADRA2A P08913 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
TACR2 P21452 2/20 0.44
SLC6A2 P23975 2/20 0.44
SLC6A4 P31645 2/20 0.44
SLC6A3 Q01959 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
SHBG P04278 1/20 0.44
TP53 P04637 1/20 0.44
CYP3A4 P08684 1/20 0.44
HSPD1 P10809 1/20 0.44
ADRB3 P13945 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28114379 0.98 HTR2A (0.52) HTR2ASIGMAR1RARBRARARARG
SCHEMBL24454689 0.98 HTR2A (0.52) HTR2ASIGMAR1RARBRARARARG
SCHEMBL530150 0.86 PNMT (0.45) SIGMAR1TP53HSD17B10GLASMN1; SMN2
SCHEMBL14402440 0.85 HTR2A (0.48) HTR2ASIGMAR1RARBRARARARG
SCHEMBL7764845 0.85 RARB (0.59) HTR2ARARBRARARARGESR1
Ammonia Solution, Strong SCHEMBL6341561 0.85 PNMT (0.44) SIGMAR1TP53HSD17B10GLASMN1; SMN2
SCHEMBL3163099 0.85 RARB (0.49) HTR2ASIGMAR1RARBRARARARG
SCHEMBL8455569 0.84 HTR2A (0.40) HTR2ASIGMAR1RARBRARARARG
SCHEMBL8455577 0.84 HTR2A (0.40) HTR2ASIGMAR1RARBRARARARG
SCHEMBL18647948 0.84 HTR2A (0.52) HTR2ASIGMAR1RARBRARARARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106232582-A Aryl and heteroaryl ether compound as ROR gamma modulators 格兰马克药品股份有限公司 2016-12-14 CN disclosed