SCHEMBL28114795

SCHEMBL28114795

COC(=O)c1cc(I)cc(N)c1Cl

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.51
GAA P10253 5/20 0.49
NQO2 P16083 6/20 0.47
KDM4E B2RXH2 6/20 0.46
CFTR P13569 3/20 0.45
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 3/20 0.45
MAPT P10636 2/20 0.45
HPGD P15428 2/20 0.45
GLA P06280 2/20 0.45
CASP1 P29466 1/20 0.45
CASP7 P55210 1/20 0.45
ATM Q13315 1/20 0.45
TSHR P16473 2/20 0.42
ALOX15 P16050 1/20 0.42
CYP3A4 P08684 1/20 0.41
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23898722 0.87 ABL1 (0.46) ABL1GAANQO2KDM4ECFTR
SCHEMBL28722488 0.84 KDM4E (0.50) ABL1GAANQO2KDM4ECFTR
SCHEMBL176841 0.82 ABL1 (0.64) ABL1GAANQO2KDM4ECFTR
SCHEMBL36846569 0.82 ABL1 (0.64) ABL1GAANQO2KDM4ECFTR
SCHEMBL28665944 0.81 KDM4E (0.59) ABL1GAANQO2KDM4ECFTR
SCHEMBL25612414 0.81 ABL1 (0.53) ABL1GAANQO2KDM4ECFTR
SCHEMBL21527283 0.79 SOS1 (0.43) ABL1GAANQO2KDM4ECFTR
SCHEMBL358224 0.79 CFTR (0.49) ABL1GAANQO2KDM4ECFTR
SCHEMBL3574538 0.79 GAA (0.49) ABL1GAANQO2KDM4ECFTR
SCHEMBL13280601 0.79 ABL1 (0.51) ABL1GAANQO2KDM4ECFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119301127-A 6-Oxo-decahydro pyrrolo [1,2-a ] [1,5] diazocine and 6-oxo-decahydro-4H-pyrrolo [2,1-d ] [1,5] thiaazacine derivatives as modulators of STAT3 and STAT6 for the treatment of cancer and inflammatory conditions 瑞克鲁迪克斯制药股份有限公司 2025-01-10 CN disclosed
CN-104812749-B Indolecarboxamide derivant as P2X7 receptor antagonist 埃科特莱茵药品有限公司 2016-12-14 CN disclosed