SCHEMBL28117572

SCHEMBL28117572

O=C(Cl)c1nccnc1Oc1cc(Cl)ccc1Cl

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 16/20 0.57
CYP2C9 P11712 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2D6 P10635 1/20 0.42
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
MEN1 O00255 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28837466 0.88 GPBAR1 (0.55) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL28117752 0.82 GPBAR1 (0.50) GPBAR1LMNAGAAHTT
SCHEMBL2329971 0.81 GPBAR1 (0.60) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL2335696 0.75 GPBAR1 (0.60) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL28117576 0.74 GPBAR1 (0.56) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL2337128 0.73 GPBAR1 (0.46) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL27885554 0.72 RHEB (0.47) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL30749510 0.71 HTR1A (0.51) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL29209321 0.71 HTR1A (0.51) GPBAR1CYP2C9CYP3A4CYP1A2CYP2C19
SCHEMBL17674836 0.70 MAPT (0.36) CYP2C9CYP1A2CYP2C19LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106317027-A Heteroaryl amide derivative and use thereof as TGR5 agonist 山东轩竹医药科技有限公司 2017-01-11 CN disclosed