SCHEMBL28118962

SCHEMBL28118962

COc1cc(OC)c(C(C)C)cc1C(=O)NN

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSD P07339 1/20 0.50
KCNK3 O14649 1/20 0.43
KCNK9 Q9NPC2 1/20 0.43
GAA P10253 3/20 0.42
POLB P06746 2/20 0.42
GFER P55789 1/20 0.42
TP53 P04637 1/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 3/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
ALDH1A1 P00352 3/20 0.40
P2RX3 P56373 2/20 0.40
P2RX2 Q9UBL9 2/20 0.40
NPSR1 Q6W5P4 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28895552 0.84 CTSD (0.61) CTSDGAAKDM4EMAPTHSD17B10
SCHEMBL23716794 0.82 CTSD (0.63) CTSDGAAPOLBKDM4EMAPT
SCHEMBL4999364 0.82 CTSD (0.39) CTSDKCNK3KCNK9POLBKDM4E
SCHEMBL382174 0.81 GAA (0.50) KCNK3KCNK9GAAPOLBGFER
SCHEMBL28292159 0.81 POLB (0.46) KCNK3KCNK9GAAPOLBGFER
SCHEMBL19818471 0.81 TP53 (0.43) KCNK3KCNK9POLBTP53KDM4E
SCHEMBL17948554 0.80 CYP3A4 (0.47) KCNK3KCNK9GAAPOLBGFER
SCHEMBL382778 0.80 HPGD (0.55) KCNK3KCNK9GAAPOLBGFER
SCHEMBL28307124 0.79 HMGCR (0.51) KCNK3KCNK9GAAPOLBGFER
SCHEMBL4999366 0.77 KDM4E (0.45) CTSDKCNK3KCNK9GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106349241-B Triazole derivative with HSP90 inhibitory activity and preparation method and application thereof 上海翰森生物医药科技有限公司 2020-04-21 CN disclosed
CN-106349241-A Triazole derivative having HSP90 (Heat Shock Protein) inhibiting activity, as well as preparation method and application of triazole derivative 上海翰森生物医药科技有限公司 2017-01-25 CN disclosed