SCHEMBL28124107

SCHEMBL28124107

CC(C)(C)OC(=O)NCC(=O)Nc1cc(Cl)c(Cl)cc1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.42
AURKB Q96GD4 2/20 0.42
AAK1 Q2M2I8 4/20 0.42
SUV39H2 Q9H5I1 2/20 0.41
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
WDR5 P61964 1/20 0.40
IDO1 P14902 2/20 0.37
MET P08581 1/20 0.36
RAF1 P04049 1/20 0.36
KDR P35968 1/20 0.36
MAP2K2 P36507 1/20 0.36
MAP2K1 Q02750 1/20 0.36
STK17B O94768 1/20 0.36
STK17A Q9UEE5 1/20 0.36
CCNB2 O95067 1/20 0.36
CCNE2 O96020 1/20 0.36
CDK1 P06493 1/20 0.36
CDK4 P11802 1/20 0.36
CCNB1 P14635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38661718 0.85 AAK1 (0.47) EGFRAURKBAAK1WDR5IDO1
SCHEMBL17132206 0.85 AAK1 (0.47) EGFRAURKBAAK1WDR5IDO1
SCHEMBL15243333 0.85 ALDH1A1 (0.44) EGFRAURKBAAK1WDR5IDO1
SCHEMBL3571997 0.84 CA12 (0.41) AAK1CA1CA2
SCHEMBL7955810 0.82 AAK1 (0.45) EGFRAURKBAAK1SUV39H2CA1
SCHEMBL38663435 0.81 AAK1 (0.48) AAK1WDR5
SCHEMBL30313179 0.81 ALDH1A1 (0.45) AAK1WDR5
SCHEMBL23731848 0.80 AAK1 (0.59) EGFRAURKBAAK1RAF1KDR
SCHEMBL22012941 0.80 AAK1 (0.64) EGFRAURKBAAK1RAF1KDR
SCHEMBL38661021 0.80 TSHR (0.45) EGFRAURKBSUV39H2CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458923-A Novel heterocyclic compound 株式会社大熊制药 2017-02-22 CN disclosed