SCHEMBL28124115

SCHEMBL28124115

COCOc1cccc(C(N)=O)c1

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 0.67
FYN P06241 2/20 0.58
TNKS O95271 1/20 0.54
PARP15 Q460N3 1/20 0.54
PARP14 Q460N5 1/20 0.54
PARP10 Q53GL7 1/20 0.54
TNKS2 Q9H2K2 1/20 0.54
PARP2 Q9UGN5 1/20 0.54
STS P08842 2/20 0.48
KMT2A Q03164 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
PRSS1 P07477 5/20 0.46
MAOB P27338 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30938023 0.85 PARP1 (0.65) PARP1TNKSPARP15PARP14PARP10
SCHEMBL202628 0.85 PARP1 (0.65) PARP1TNKSPARP15PARP14PARP10
SCHEMBL30442255 0.85 MAOB (0.62) KMT2AMAOB
SCHEMBL3148484 0.85 KMT2A (0.66) KMT2A
SCHEMBL3151885 0.85 MAOB (0.62) KMT2AMAOB
SCHEMBL6356224 0.83 KMT2A (0.47) PARP1FYNKMT2ACES2CES1
SCHEMBL3069825 0.83 MRGPRX4 (0.56) KMT2ACES2CES1
SCHEMBL2705442 0.83 PARP1 (0.66) PARP1TNKSPARP15PARP14PARP10
SCHEMBL3161225 0.83 SMPD1 (0.49) PARP1KMT2A
SCHEMBL1548903 0.82 KMT2A (0.50) PARP1KMT2ACES2CES1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458892-B It is used to prepare a times improved method for carcinomycin prodrug 斯索恩生物制药有限公司 2019-10-18 CN disclosed
CN-106458892-A Improved process for making duocarmycin prodrugs 斯索恩生物制药有限公司 2017-02-22 CN disclosed