SCHEMBL28124192

SCHEMBL28124192

CCON(CCOC)C1CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.42
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
PIK3CD O00329 1/20 0.36
GPR119 Q8TDV5 3/20 0.34
USP2 O75604 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
USP30 Q70CQ3 2/20 0.34
NAMPT P43490 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21494393 0.81 NR1H2 (0.46) NR1H2DDB1CRBNPIK3CDGPR119
SCHEMBL28124182 0.77 NR1H2 (0.48) NR1H2DDB1CRBNGPR119USP2
SCHEMBL17910144 0.77 NR1H2 (0.46) NR1H2DDB1CRBNPIK3CDGPR119
SCHEMBL24680916 0.74 USP30 (0.48) DDB1CRBNPIK3CDGPR119USP30
SCHEMBL31208730 0.74 USP30 (0.48) DDB1CRBNPIK3CDGPR119USP30
SCHEMBL24680917 0.74 USP30 (0.48) DDB1CRBNPIK3CDGPR119USP30
SCHEMBL22989452 0.73 NR1H2 (0.49) NR1H2DDB1CRBNGPR119USP2
SCHEMBL24033629 0.73 NR1H2 (0.44) NR1H2DDB1CRBNPIK3CDGPR119
SCHEMBL24161826 0.72 NR1H2 (0.51) NR1H2DDB1CRBNGPR119USP2
SCHEMBL20896506 0.72 NR1H2 (0.43) NR1H2DDB1CRBNPIK3CDGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459034-B Carbostyril derivative as fibroblast growth factor acceptor inhibitor 普林斯匹亚生物制药公司 2018-01-12 CN disclosed
CN-106459034-A Quinolone derivatives as fibroblast growth factor receptor inhibitors 普林斯匹亚生物制药公司 2017-02-22 CN disclosed