SCHEMBL28124221

SCHEMBL28124221

[CH2]CNc1nc(N)nc2[nH]ncc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
CDK2 P24941 2/20 0.42
ALDH1A1 P00352 2/20 0.40
CYP1A2 P05177 2/20 0.38
PDPK1 O15530 1/20 0.38
HTR2A P28223 3/20 0.37
NLRP3 Q96P20 1/20 0.37
LMNA P02545 1/20 0.37
RET P07949 1/20 0.37
PI4KA P42356 1/20 0.37
XDH P47989 1/20 0.37
LRRK2 Q5S007 1/20 0.37
PI4K2B Q8TCG2 1/20 0.37
PI4K2A Q9BTU6 1/20 0.37
PI4KB Q9UBF8 1/20 0.37
POLB P06746 1/20 0.37
HTR2C P28335 3/20 0.36
RECQL P46063 1/20 0.35
SLC29A1 Q99808 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31706902 0.77 PDPK1 (0.58) ADORA2AADORA1CDK2ALDH1A1PDPK1
SCHEMBL129637 0.77 PDPK1 (0.58) ADORA2AADORA1CDK2ALDH1A1PDPK1
SCHEMBL14561714 0.75 ADORA2A (0.43) ADORA2AADORA1CDK2ALDH1A1CYP1A2
SCHEMBL1014920 0.72 XDH (0.55) ADORA2AADORA1CDK2ALDH1A1PDPK1
SCHEMBL29487078 0.72 XDH (0.55) ADORA2AADORA1CDK2ALDH1A1PDPK1
Benzene SCHEMBL25427466 0.69 RET (0.52) ADORA2AADORA1CDK2PDPK1RET
SCHEMBL2629520 0.69 ADORA2A (0.47) ADORA2AADORA1CDK2ALDH1A1PDPK1
SCHEMBL19891462 0.69 ADORA2A (0.47) ADORA2AADORA1CDK2ALDH1A1PDPK1
SCHEMBL341706 0.69 ADORA2A (0.47) ADORA2AADORA1CDK2ALDH1A1LMNA
SCHEMBL888387 0.69 ADORA2A (0.47) ADORA2AADORA1CDK2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459012-A Quinazolinone derivatives as phosphatidylinositol 3-kinase inhibitors 吉利德科学公司 2017-02-22 CN claimed