SCHEMBL28127686

SCHEMBL28127686

FC(F)(F)c1cc(Cn2cccn2)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.51
MAPT P10636 1/20 0.51
IDO1 P14902 2/20 0.47
KCNN4 O15554 3/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
HTT P42858 1/20 0.45
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
OPRK1 P41145 2/20 0.43
NOTUM Q6P988 1/20 0.43
FAAH O00519 1/20 0.42
ADORA2B P29275 1/20 0.42
MEN1 O00255 1/20 0.41
TSHR P16473 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13122997 0.83 HTT (0.45) GAAMAPTHDAC1HDAC6HTT
SCHEMBL18235820 0.82 GAA (0.59) GAAMAPTHDAC1HDAC6HTT
SCHEMBL28839857 0.81 HTT (0.46) GAAMAPTHDAC1HDAC6HTT
SCHEMBL17310038 0.81 GAA (0.55) GAAMAPTHDAC1HDAC6HTT
SCHEMBL13122968 0.80 HTT (0.42) GAAMAPTHDAC1HDAC6HTT
SCHEMBL28127687 0.80 GAA (0.48) GAAMAPTKCNN4HDAC1HDAC6
SCHEMBL14822758 0.79 MAPT (0.55) GAAMAPTHDAC1HDAC6HTT
SCHEMBL28149998 0.77 CA12 (0.51) GAAMAPTHDAC1HDAC6HTT
SCHEMBL16969000 0.77 IDO1 (0.47) IDO1KCNN4OPRK1FAAHADORA2B
SCHEMBL17316747 0.76 L3MBTL1 (0.52) IDO1KCNN4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106414429-A Pyrazole compounds and their use as T-type calcium channel blockers 埃科特莱茵药品有限公司 2017-02-15 CN disclosed