Reserpine

Reserpine

SCHEMBL28129

C1=CC2C3C=CC(C3)C2C1.COC(=O)[C@H]1[C@H]2C[C@@H]3c4[nH]c5cc(OC)ccc5c4CCN3C[C@H]2C[C@@H](OC(=O)c2cc(OC)c(OC)c(OC)c2)[C@@H]1OC

nearest known ligand 0.84

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SLC18A2

The experimentally established mechanism targets of Reserpine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC18A2 known ✓ Q05940 1/20 0.84
MEN1 O00255 13/20 0.84
KMT2A Q03164 13/20 0.84
KDM4E B2RXH2 10/20 0.84
TDP1 Q9NUW8 7/20 0.84
TSHR P16473 6/20 0.84
MAPT P10636 6/20 0.84
HBB P68871 5/20 0.84
ALDH1A1 P00352 5/20 0.84
CYP3A4 P08684 4/20 0.84
USP2 O75604 4/20 0.84
CASP1 P29466 4/20 0.84
ALOX15 P16050 3/20 0.84
KCNH2 Q12809 3/20 0.84
CASP7 P55210 3/20 0.84
HSD17B10 Q99714 2/20 0.84
ADORA3 P0DMS8 2/20 0.84
OPRM1 P35372 2/20 0.84
OPRK1 P41145 2/20 0.84
CYP1A2 P05177 2/20 0.84

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Reserpine SCHEMBL20402680 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL14379427 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Isoreserpine SCHEMBL731599 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL12732449 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL5372164 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL8262666 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL4562878 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL15385127 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL22002247 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR
Reserpine SCHEMBL1172973 0.92 MEN1 (1.00) MEN1KMT2AKDM4ETDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3677438-B1 PNEUMATIC TIRE BRIDGESTONE CORP (JP) 2023-11-15 EP claimed
EP-2759400-B1 LAMINATED BODY, LAMINATED BOARD, MULTI-LAYER LAMINATED BOARD, PRINTED WIRING BOARD, AND PRODUCTION METHOD FOR LAMINATED BOARD HITACHI CHEMICAL CO LTD (JP) 2020-04-15 EP claimed
EP-3359398-B1 TIRE FOR AGRICULTURAL VEHICLE MICHELIN & CIE (FR) 2019-09-04 EP claimed
EP-3126155-B1 RUBBER COMPOSITION COMPRISING AN AROMATIC DICYCLOPENTADIENE RESIN MICHELIN & CIE (FR) 2019-07-24 EP claimed
EP-2388299-B1 Infrared absorbing composition, infrared absorbing ink, recorded article, image recording method, and image detecting method FUJIFILM CORP (JP) 2017-12-06 EP claimed
WO-2017060633-A1 TIRE FOR AGRICULTURAL VEHICLE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2017-04-13 WO claimed
EP-3126155-A1 RUBBER COMPOSITION COMPRISING AN AROMATIC DICYCLOPENTADIENE RESIN Compagnie Générale des Etablissements Michelin (FR) 2017-02-08 EP claimed
WO-2015150542-A1 RUBBER COMPOSITION COMPRISING AN AROMATIC DICYCLOPENTADIENE RESIN COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2015-10-08 WO claimed
EP-1215248-B1 Process for producing a resin molded product SHINETSU CHEMICAL CO (JP) 2009-04-29 EP claimed
EP-1667562-B1 COMPOSITE ARTICLE AND METHOD OF MANUFACTURE KOHLER MIRA LTD (GB) 2008-11-19 EP claimed
EP-1314802-B1 Temperature-sensitive color-changeable composite fiber PILOT INK CO LTD (JP) 2007-03-28 EP claimed
EP-1386724-B1 Barrier coat for open tool molding GEN MOTORS CORP (US) 2006-10-11 EP claimed
EP-1566546-B1 Scroll compressor and refrigerating system using ammonia HITACHI AIR CONDITIONING SYS (JP) 2006-08-02 EP claimed
EP-1352008-B1 EPOXY RESIN COMPOSITION FOR SEMICONDUCTOR ENCAPSULATION RESOLUTION RES NEDERLAND BV (NL) 2005-06-29 EP claimed
EP-1228119-B1 HIGH PERFORMANCE POLYETHERESTER CONTAINING LAMINATING RESIN COMPOSITIONS REICHHOLD INC (US) 2003-11-19 EP claimed
EP-0065195-B1 BINDER FOR TOLUENE DEEP PRINTING INKS BASF Aktiengesellschaft (DE) 1984-03-14 EP claimed
EP-4037919-A1 RUBBER COMPOSITION FOR A LARGE-SIZED TIRE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2022-08-10 EP disclosed
WO-2021064317-A1 RUBBER COMPOSITION FOR A LARGE-SIZED TIRE COMPAGNIE GENERALE DES ETABLISSEMENTS MICHELIN (FR) 2021-04-08 WO disclosed
WO-2003072357-A2 METALLISABLE, ORIENTED, MULTILAYER POLYOLEFIN FILM UCB, S.A. (BE) 2003-09-04 WO disclosed
WO-2002090090-A1 METHOD OF PRODUCING A MOULDED ARTICLE COURTNEY WYNDHAM JAMES (GB) 2002-11-14 WO disclosed