SCHEMBL28136286

SCHEMBL28136286

CCC(=O)Oc1cc([N+](=O)[O-])c(F)cc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.43
RECQL P46063 2/20 0.43
MAPT P10636 4/20 0.41
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
VCP P55072 1/20 0.40
HTT P42858 1/20 0.39
KMT2A Q03164 5/20 0.38
LMNA P02545 4/20 0.38
MEN1 O00255 3/20 0.38
RAB9A P51151 1/20 0.36
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36
PDGFRA P16234 1/20 0.36
FLT1 P17948 1/20 0.36
FGFR3 P22607 1/20 0.36
KDR P35968 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27972345 0.85 RECQL (0.42) RECQLMAPTALDH1A1SMN1; SMN2VCP
SCHEMBL28405700 0.85 MEN1 (0.40) RECQLMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL1098698 0.84 MAPT (0.39) RECQLMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL29739365 0.84 MAPT (0.39) RECQLMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL28405701 0.84 TSHR (0.41) RECQLMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL28136377 0.84 ITGB1 (0.40) ACHEMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL29739370 0.79 MAPT (0.43) RECQLMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL187546 0.77 ALDH1A1 (0.49) MAPTALDH1A1HTTESPL1KDM4E
SCHEMBL29739457 0.77 ALDH1A1 (0.49) MAPTALDH1A1HTTESPL1KDM4E
SCHEMBL3475943 0.77 TDP1 (0.43) MAPTALDH1A1SMN1; SMN2HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106573897-B Benzimidazol-2-amines as mIDH1 inhibitors 拜耳制药股份公司 2019-09-24 CN disclosed
CN-106573897-A Benzimidazol-2-amines as MiDH1 inhibitors 拜耳制药股份公司 2017-04-19 CN disclosed